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[18F]fluoro-benziodoxole: a no-carrier-added electrophilic fluorinating reagent. Rapid, simple radiosynthesis, purification and application for fluorine-18 labelling
Stockholm Univ, Dept Organ Chem, SE-10691 Stockholm, Sweden.
Uppsala University, Disciplinary Domain of Medicine and Pharmacy, Faculty of Pharmacy, Department of Medicinal Chemistry, Preparative Medicinal Chemistry.
Stockholm Univ, Dept Organ Chem, SE-10691 Stockholm, Sweden;Karolinska Inst, AstraZeneca PET Ctr, SE-17176 Stockholm, Sweden.
Stockholm Univ, Dept Organ Chem, SE-10691 Stockholm, Sweden.ORCID iD: 0000-0002-8834-9834
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2018 (English)In: Chemical Communications, ISSN 1359-7345, E-ISSN 1364-548X, Vol. 54, no 34, p. 4286-4289Article in journal (Refereed) Published
Abstract [en]

Operationally simple radiosynthesis and purification of [F-18]fluoro-benziodoxole was developed starting from a cyclotron produced [F-18]F- precursor, [F-18]TBAF, and tosyl-benziodoxole. The synthetic utility of [F-18]fluoro-benziodoxole was demonstrated by electrophilic fluorocyclization of o-styrilamides proceeding with high RCC (typically 50-90%) and high molar activity (up to 396 GBq mol(-1)).

Place, publisher, year, edition, pages
2018. Vol. 54, no 34, p. 4286-4289
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Organic Chemistry
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URN: urn:nbn:se:uu:diva-354948DOI: 10.1039/c8cc00526eISI: 000430935200013PubMedID: 29632936OAI: oai:DiVA.org:uu-354948DiVA, id: diva2:1223529
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VINNOVASwedish Research CouncilAvailable from: 2018-06-25 Created: 2018-06-25 Last updated: 2018-06-25Bibliographically approved

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